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The Pharmaceutical Journal Vol 265 No 7104 p63
July 8, 2000 Forum

International symposium on atherosclerosis

Inhibiting cholesterol absorption

The reports on this and the next page are from the XIIth International Symposium on Atherosclerosis which was held in Stockholm on June 25-29
Reports include: Bayer tests cerivastatin in renal disease; New cancer drugs might also find use in heart disease; HDL-mimetics; Gene therapy trial in peripheral vascular disease; Beta-blocker benefit in atherosclerosis?; Benefit shown for treating lipid disorders in patients with diabetes

Several pharmaceutical companies are developing new lipid lowering drugs that act by inhibiting cholesterol absorption. Dr H. Davis, from Schering Plough, US, discussed his company's compound ezetimibe. He said that the drug inhibited both dietary and biliary cholesterol absorption. Dr Davis reported studies in which ezetimibe inhibited the normal rise in LDL cholesterol in monkeys fed a western diet, without affecting HDL or triglyceride levels. He suggested that combining the drug with a statin might give additional lowering of LDL. Hepatic synthesis of cholesterol was increased with ezetimibe but this could be blocked by statin therapy.